Dactinomycin
Synonyms
Ac-De
Actinomycin
Actinomycin D
Cosmegen
Cosmegen Lyovac
Lemery Brand of Dactinomycin
Lyovac, Cosmegen
Lyovac-Cosmegen
MSD Brand of Dactinomycin
Meractinomycin
Merck Brand of Dactinomycin
Merck Frosst Brand of Dactinomycin
Merck Sharp & Dohme Brand of Dactinomycin
A compound composed of a two CYCLIC PEPTIDES attached to a phenoxazine that is derived from STREPTOMYCES parvullus. It binds to DNA and inhibits RNA synthesis (transcription), with chain elongation more sensitive than initiation, termination, or release. As a result of impaired mRNA production, protein synthesis also declines after dactinomycin therapy. (From AMA Drug Evaluations Annual, 1993, p2015)